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Title:Identification of furin protease small-molecule inhibitor with a 1,3-thiazol-2-ylaminosulfonyl scaffold
Authors:ID Kolarič, Anja (Author)
ID Ravnik, Vid (Author)
ID Štumpf Horvat, Sara (Author)
ID Jukič, Marko (Author)
ID Bren, Urban (Author)
Files:.pdf pharmaceuticals-18-00273_(1).pdf (6,26 MB)
MD5: 61590D80702F0B474D38342A80F73F47
 
Language:English
Work type:Article
Typology:1.01 - Original Scientific Article
Organization:FKKT - Faculty of Chemistry and Chemical Engineering
Keywords:computer-assisted drug design, CADD, computer-assisted drug design, furin inhibitors, protease inhibitors, antivirals, protease inhibitors, furin assay, antiviral drug design
Publication status:Published
Publication version:Version of Record
Submitted for review:09.02.2025
Article acceptance date:15.02.2025
Publication date:19.02.2025
Year of publishing:2025
Number of pages:15 str.
Numbering:Vol. 18, no. 2, [Article no.] 273
PID:20.500.12556/DKUM-92201 New window
UDC:577
ISSN on article:1424-8247
COBISS.SI-ID:227126787 New window
DOI:10.3390/ph18020273 New window
Copyright:© 2025 by the authors
Publication date in DKUM:20.03.2025
Views:142
Downloads:8
Metadata:XML DC-XML DC-RDF
Categories:Misc.
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Record is a part of a journal

Title:Pharmaceuticals
Shortened title:Pharmaceuticals
Publisher:MDPI, Molecular Diversity Preservation International
ISSN:1424-8247
COBISS.SI-ID:517582617 New window

Document is financed by a project

Funder:ARIS - Slovenian Research and Innovation Agency
Project number:J1-2471-2020
Name:Kemijska karcinogeneza: Mehanistični vpogled

Funder:ARIS - Slovenian Research and Innovation Agency
Project number:P2-0046-2019
Name:Separacijski procesi in produktna tehnika

Funder:ARIS - Slovenian Research and Innovation Agency
Project number:L2-3175-2021
Name:Napredna ekstrakcija in formulacija funkcionalnih taninskih prahranskih dopolnil z blagodejnimi zdravstvenimi učinki

Funder:ARIS - Slovenian Research and Innovation Agency
Project number:J4-4633-2023
Name:Razumevanje mehanizmov in preprečevanje agregacije biofarmacevtskih proteinov

Funder:ARIS - Slovenian Research and Innovation Agency
Project number:J1-4398-2022
Name:Kemijska karcinogeneza in nevrodegeneracija: Molekularni mehanizem vpliva mikrovalovnega sevanja

Funder:ARIS - Slovenian Research and Innovation Agency
Project number:L2-4430-2022
Name:Proizvodnja, izolacija in formulacija zdravju koristnih substanc iz Helichrysum Italicum za uporabo v kozmetični industriji

Funder:ARIS - Slovenian Research and Innovation Agency
Project number:J3-4498-2022
Name:Multi-omska raziskava signalne poti NFkB pri multipli sklerozi

Funder:ARIS - Slovenian Research and Innovation Agency
Project number:J7-4638-2022
Name:Načrtovanje selektivnih katalitskih postopkov pretvorbe CO2 v etanol – UliSess

Funder:ARIS - Slovenian Research and Innovation Agency
Project number:J1-4414-2022
Name:ProBiS-Fold pristop za določanje vezavnih mest za celoten strukturni človeški proteom pri odkrivanju zdravil

Funder:ARIS - Slovenian Research and Innovation Agency
Project number:J3-4497-2022
Name:Neinvazivni multi-omski biooznačevalci v podtipih imunskih celic za personalizirano zdravljenje otroške astme in molekularni mehanizmi neodzivnosti na inhalacijske kortikosteroide

Funder:ARIS - Slovenian Research and Innovation Agency
Project number:P2-0438-2022
Name:Optični kemijski/bio senzorski sistemi (OPTISENS)

Funder:ARIS - Slovenian Research and Innovation Agency
Project number:J1-50034-2023
Name:Knjižnica korelacij med vezavnimi vzorci opioidov in njihovimi neželenimi stranskimi učinki

Funder:ARIS - Slovenian Research and Innovation Agency
Project number:J7-50043-2023
Name:Mutacijska platforma koronavirusnih terapevtskih tarč za študij vpliva mutacij na učinkovitost in izbiro zdravil ter načrtovanje novih pan-koronavirusnih zaviralcev

Funder:ARIS - Slovenian Research and Innovation Agency
Project number:Z1-50021-2024
Name:Uravnoteženo dvojno ciljanje hibridov novih zaviralcev bakterijske topoizomeraze-fluorokinolonov (NBTI-FQ) kot inovativen pristop v boju proti bakterijski odpornosti

Funder:ARIS - Slovenian Research and Innovation Agency
Project number:P1-0403-2019
Name:Računsko intenzivni kompleksni sistemi

Funder:ARIS - Slovenian Research and Innovation Agency
Project number:I0-E015-2024
Name:Izvajanje mednarodnega infrastrukturnega projekta BBMRI

Licences

License:CC BY 4.0, Creative Commons Attribution 4.0 International
Link:http://creativecommons.org/licenses/by/4.0/
Description:This is the standard Creative Commons license that gives others maximum freedom to do what they want with the work as long as they credit the author.

Secondary language

Language:Slovenian
Keywords:zdravila, inhibitorji, protivirusi


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